Methylarginine Targeting Chimeras for Lysosomal Degradation of Intracellular Proteins

  • Methylarginine degrons are a widespread signal for intracellular protein delivery to lysosomes
  • MrTAC is a first-in-class lysosomal degrader
  • Methyl-driven lysosomal proteolysis expands the scope of current proximity inducing modalities to new families of undruggable targe